Nastorazepide (hemicalcium), CAS [[343326-69-2]] Preis auf Anfrage
Artikelnummer:
MCE-HY-14575
Hersteller Artikelnummer:
HY-14575
Alternativnummer:
MCE-HY-14575-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Alternative Synonym:
Z-360 (hemicalcium)
Nastorazepide (Z-360) hemicalcium is an orally active 1,5-benzodiazepine derivative and gastrin/CCK-2 receptor antagonist. Nastorazepide hemicalcium inhibits the specific binding of [3H]CCK-8 to the human CCK-2 receptor with a Ki value of 0.47 nM. Nastorazepide hemicalcium inhibits IL-1beta, ephrin B1, VEGF, and HIF-1alpha, reduces Akt and NR2B phosphorylation. Nastorazepide hemicalcium has antitumor activity against pancreatic cancer. Nastorazepide hemicalcium inhibits colorectal cancer liver metastasis and relieves pain[1][2][3][4][5][6][7].
