TIY-7, CAS [[2846435-83-2]] Preis auf Anfrage
Artikelnummer:
MCE-HY-146755
| Artikelname: |
TIY-7, CAS [[2846435-83-2]] Preis auf Anfrage |
| Artikelnummer: |
MCE-HY-146755 |
| Hersteller Artikelnummer: |
HY-146755 |
| Alternativnummer: |
MCE-HY-146755-1UNIT |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| TIY-7 is a selective and orally active tropomyosin receptor kinase (TRK) inhibitor. TIY-7 shows enzyme inhibitory activity with IC50s of 2.9, 1.1, 0.7, 0.8, 0.8, 0.2 nM for TRKA, TRKAG595R, TRKAG667C, TRKAF589L, TRKCG623R, TRKCG696A, respectively. TIY-7 shows anti-tumor potency in mouse xenograft model[1]. |
| Molekulargewicht: |
446.40 |
| CAS Nummer: |
[2846435-83-2] |
| Formel: |
C21H18F4N6O |
| Target-Kategorie: |
Trk Receptor |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |