Desmethylazelastine is a main active metabolite of Azelastine that is oxidatively metabolized by the cytochrome P450 enzyme system with a protein binding rate of 97% and an elimination half-life of 54 hours. Azelastine is an orally active, selective and high-affinity histamine H1-receptor antagonist. Azelastine can be used in studies of allergic rhinitis, asthma, diabetic hyperlipidemic and SARS-CoV-2[1][2][3][4][5].
Molekulargewicht:
367.87
CAS Nummer:
[47491-38-3]
Formel:
C21H22ClN3O
Target-Kategorie:
Drug Metabolite
Anwendungsbeschreibung:
MCE Product type: Reference compound
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