ERD-3111, CAS [[2832865-25-3]]

Artikelnummer: MCE-HY-149480
Artikelname: ERD-3111, CAS [[2832865-25-3]]
Artikelnummer: MCE-HY-149480
Hersteller Artikelnummer: HY-149480
Alternativnummer: MCE-HY-149480-10MG,MCE-HY-149480-5MG,MCE-HY-149480-25MG,MCE-HY-149480-1MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
ERD-3111 (Compound 44) is an orally active PROTAC ERalpha degrader (DC50: 0.5 nM). ERD-3111 inhibits tumor growth in the parental MCF-7 xenograft model with wild-type ER and two clinically relevant ESR1 mutated mice model. ERD-3111 can be used in the research of ER+ breast cancer[1].
Molekulargewicht: 854.89
Reinheit: 98.72
CAS Nummer: [2832865-25-3]
Formel: C45H46F4N8O5
Target-Kategorie: Estrogen Receptor/ERR,PROTACs
Anwendungsbeschreibung: Reference compound