BD-9136 is a potent and highly selective BRD4 PROTAC depressant. BD-9136 has low-nanomolar degradation potencies against BRD4 , and its degradation selectivity for BRD4 is 1000 times that of BRD2 and BRD3 proteins. BD-9136 has antitumor activity[1].(Pink: Desmethyl-QCA276 (HY-44103), Black: 3-(2-(4-Methylpiperazin-1-yl)ethyl)azetidin-3-ol, Blue: Thalidomide-4-OH (HY-103596))
Molekulargewicht:
824.95
Reinheit:
98.81
CAS Nummer:
[3037514-38-5]
Formel:
C44H44N10O5S
Target-Kategorie:
Epigenetic Reader Domain,PROTACs
Anwendungsbeschreibung:
MCE Product type: Reference compound
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