EM127, CAS [[1886879-71-5]]

Produktübersicht

• Artikelname: EM127, CAS [[1886879-71-5]]
• Artikelnummer: MCE-HY-151379
• Hersteller Artikelnummer: HY-151379
• Alternativnummer: MCE-HY-151379-10MMX1ML,MCE-HY-151379-50MG,MCE-HY-151379-25MG,MCE-HY-151379-10MG,MCE-HY-151379-100MG,MCE-HY-151379-5MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

EM127 (compound 11c) is a SMYD3 covalent inhibitor with high selectivity, high affinity (KD=13 µM) and site-specificity. EM127 effectively inhibits ERK1/2 phosphorylation and reduces transcriptional regulation of SMYD3 target genes. EM127 effectively and prolongedly impairs methyltransferase activity. EM127 can be used in cancer research, particularly in SMYD3 positive tumours[1].

Produkteigenschaften

• Molekulargewicht: 311.76
• Reinheit: 99.94
• CAS Nummer: [1886879-71-5]
• Formel: C14H18ClN3O3
• Target-Kategorie: Histone Methyltransferase

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound