Bemcentinib, CAS [[1037624-75-1]]

Artikelnummer: MCE-HY-15150
Artikelname: Bemcentinib, CAS [[1037624-75-1]]
Artikelnummer: MCE-HY-15150
Hersteller Artikelnummer: HY-15150
Alternativnummer: MCE-HY-15150-200MG,MCE-HY-15150-5MG,MCE-HY-15150-10MG,MCE-HY-15150-100MG,MCE-HY-15150-10MMX1ML,MCE-HY-15150-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: R428, BGB324
Bemcentinib (R428) is a selective and orally active Axl inhibitor with an IC50 of 14 nM. Bemcentinib retards cancer cell migration and invasion. Bemcentinib exhibits >100-fold selectivity for Axl versus Abl and 50- and >100-fold selectivity over TAM family kinases Mer and Tyro3, respectively, in cells. Bemcentinib blocks tumor spread and prolongs survival in models of metastatic breast cancer[1][2].
Molekulargewicht: 506.64
Reinheit: 99.92
CAS Nummer: [1037624-75-1]
Formel: C30H34N8
Target-Kategorie: TAM Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound