MRS542 is a nucleoside A3 AR antagonist with a pKi of 8.74. MRS542 also acts as a partial agonist (pEC50 = 7.76) in promoting beta-arrestin translocation. MRS542 can be converted into an agonist by LUF6000 (HY-13236). MRS542 can be used for cardiovascular disease research[1][2].
Molekulargewicht:
517.71
CAS Nummer:
[163152-31-6]
Formel:
C17H17ClIN5O4
Target-Kategorie:
Adenosine Receptor,Arrestin
Anwendungsbeschreibung:
MCE Product type: Reference compound
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