DDO-2213, CAS [[2378768-36-4]]

Artikelnummer: MCE-HY-153331
Artikelname: DDO-2213, CAS [[2378768-36-4]]
Artikelnummer: MCE-HY-153331
Hersteller Artikelnummer: HY-153331
Alternativnummer: MCE-HY-153331-5MG,MCE-HY-153331-10MG,MCE-HY-153331-100MG,MCE-HY-153331-25MG,MCE-HY-153331-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
DDO-2213 is an orally active and potent WDR5-MLL1 inhibitor, with an IC50 of 29 nM and a Kd value of 72.9 nM for the WDR5 protein. DDO-2213 selectively inhibits MLL (mixed lineage leukemia) histone methyltransferase activity and the proliferation of MLL translocation-harboring cells. DDO-2213 can be used for MLL fusion leukemia research[1].
Molekulargewicht: 483.97
Reinheit: 98.84
CAS Nummer: [2378768-36-4]
Formel: C24H27ClFN7O
Target-Kategorie: WDR5
Anwendungsbeschreibung: Reference compound