Gintemetostat, CAS [[2604513-16-6]]

Produktübersicht

• Artikelname: Gintemetostat, CAS [[2604513-16-6]]
• Artikelnummer: MCE-HY-154812
• Hersteller Artikelnummer: HY-154812
• Alternativnummer: MCE-HY-154812-100MG,MCE-HY-154812-5MG,MCE-HY-154812-10MG,MCE-HY-154812-25MG,MCE-HY-154812-50MG,MCE-HY-154812-10MMX1ML
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: KTX-1001

Produktbeschreibung

Gintemetostat is an orally available, highly specific NSD2/MMSET histone methyltransferase inhibitor with human NSD2 IC50 values ranging 0.460-2.17 nM and NSD2 SET domain IC50 of 2.32 nM and Kd values ranging 6.3-70.4 nM[1][4].Gintemetostat reduces H3K36me2 levels, impairs multiple myeloma cell adhesion and colony formation, enhances cytotoxicity, boosts T-cell activation, and sensitizes resistant multiple myeloma cells to other agents[1][2][6].Gintemetostat can be used for the research of multiple myeloma and relapsed and refractory multiple myeloma[1][2][3][4][5][6].

Produkteigenschaften

• Molekulargewicht: 546.52
• Reinheit: 99.81
• CAS Nummer: [2604513-16-6]
• Formel: C25H26F4N8O2
• Target-Kategorie: CD44,Histone Methyltransferase

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound