PROTAC TG2 degrader-2 (compound 7) is a selective, competitive degrader targeting Transglutaminase 2 (TG2), with Kd > 100 µM. PROTAC TG2 degrader-2 inhibits the cell migration and decreases the level of TG2 in ovarian cancer cells. PROTAC TG2 degrader-2 can be used for ovarian cancer study[1].
Molekulargewicht:
876.08
Reinheit:
99.15
Formel:
C47H57N9O6S
Target-Kategorie:
Glutaminase,PROTACs
Anwendungsbeschreibung:
MCE Product type: Reference compound
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