Ceritinib (mesylate), CAS [[2055376-74-2]] Preis auf Anfrage

Artikelnummer: MCE-HY-15656B
Artikelname: Ceritinib (mesylate), CAS [[2055376-74-2]] Preis auf Anfrage
Artikelnummer: MCE-HY-15656B
Hersteller Artikelnummer: HY-15656B
Alternativnummer: MCE-HY-15656B-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: LDK378 (mesylate)
Ceritinib (LDK378) mesylate is a selective, orally bioavailable, and ATP-competitive ALK tyrosine kinase inhibitor with an IC50 of 200 pM. Ceritinib mesylate also inhibits IGF-1R, InsR, and STK22D with IC50 values of 8, 7, and 23 nM, respectively. Ceritinib mesylate shows great antitumor potency[1][2].
Molekulargewicht: 750.35
CAS Nummer: [2055376-74-2]
Formel: C30H44ClN5O9S3
Target-Kategorie: Anaplastic lymphoma kinase (ALK),IGF-1R,Insulin Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound