Ceritinib (mesylate), CAS [[2055376-74-2]] Preis auf Anfrage
Artikelnummer:
MCE-HY-15656B
Hersteller Artikelnummer:
HY-15656B
Alternativnummer:
MCE-HY-15656B-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Alternative Synonym:
LDK378 (mesylate)
Ceritinib (LDK378) mesylate is a selective, orally bioavailable, and ATP-competitive ALK tyrosine kinase inhibitor with an IC50 of 200 pM. Ceritinib mesylate also inhibits IGF-1R, InsR, and STK22D with IC50 values of 8, 7, and 23 nM, respectively. Ceritinib mesylate shows great antitumor potency[1][2].