CRT0066101 (trihydrochloride), CAS [[1781742-22-0]] Preis auf Anfrage
Artikelnummer:
MCE-HY-15698B
Hersteller Artikelnummer:
HY-15698B
Alternativnummer:
MCE-HY-15698B-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
CRT0066101 trihydrochloride is the trihydrochloride salt form of CRT0066101 (HY-15698). CRT0066101 trihydrochloride is an orally active PKD inhibitor with IC50 values of 1 nM, 2.5 nM and 2 nM for PKD1, PKD2, and PKD3, respectively. CRT0066101 trihydrochloride is also an inhibitor for PIM2 with an IC50 of ~135.7 nM. CRT0066101 trihydrochloride exhibits anti-inflammatory activity in mice LPS (HY-D1056)-induced lung injury models, and has anticancer effects[1][2][3].
Molekulargewicht:
447.79
CAS Nummer:
[1781742-22-0]
Formel:
C18H25Cl3N6O
Target-Kategorie:
Apoptosis,Pim,PKD
Anwendungsbeschreibung:
MCE Product type: Reference compound
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