Brexpiprazole (hydrochloride), CAS [[913612-38-1]] Preis auf Anfrage
Artikelnummer:
MCE-HY-15780A
Hersteller Artikelnummer:
HY-15780A
Alternativnummer:
MCE-HY-15780A-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Alternative Synonym:
OPC-34712 (hydrochloride)
Brexpiprazole (OPC-34712) hydrochloride, an atypical orally active antipsychotic agent, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole hydrochloride is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole hydrochloride also shows potent antagonist activity at human noradrenergic alpha1B (Ki=0.17 nM) and alpha2C receptors (Ki=0.59 nM)[1][2].
