MR24, a G-5555 (HY-19635) derivative, is a mammalian STE20-like (MST) kinase inhibitor. MR24 shows selectively to MST3/4 over MST1/2, with EC50 values of 57 and 583 nM, respectively. MR24 induces G1 phase cell cycle arrest. MR24 can be used for cancer research, such as breast, liver and lung cancers[1].
Molekulargewicht:
509.00
CAS Nummer:
[3056814-89-9]
Formel:
C26H29ClN6O3
Target-Kategorie:
Hippo (MST)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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