CBPD-409, CAS [[3037549-86-0]]

Produktübersicht

• Artikelname: CBPD-409, CAS [[3037549-86-0]]
• Artikelnummer: MCE-HY-158113
• Hersteller Artikelnummer: HY-158113
• Alternativnummer: MCE-HY-158113-5MG,MCE-HY-158113-10MG,MCE-HY-158113-1MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

CBPD-409 is an orally active PROTAC degrader for CBP/p300, with DC50 of 0.2-0.4 nM. CBPD-409 exhibits antiproliferative effects in AR+ prostate cancer cell lines VCaP, LNCaP and 22Rv1, with IC50s of 1.2-2.0 nM. CBPD-409 exhibits antitumor efficacy (Red: CBP inhibitor GNE049 (HY-108435), Blue: CRBN/cullin 4A Thalidomide (HY-14658), Black: Linker)[1].

Produkteigenschaften

• Molekulargewicht: 862.97
• Reinheit: 99.38
• CAS Nummer: [3037549-86-0]
• Formel: C46H52F2N10O5
• Target-Kategorie: Histone Acetyltransferase,PROTACs

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound