VRK1/CK1-IN-1 (compound 36) is a dual VRK1 and CK1 family inhibitor, with a Ki of 37.9 nM against human VRK1, 8.3 nM against human CK1delta, and 7.8 nM against human CK1epsilon. VRK1/CK1-IN-1 exhibits extremely low activity against VRK2. VRK1/CK1-IN-1 can be used in studies related to p53-deficient tumors[1].
Molekulargewicht:
416.38
Reinheit:
98.69
CAS Nummer:
[3050772-20-5]
Formel:
C19H18F2N6O3
Target-Kategorie:
Casein Kinase,VRK
Anwendungsbeschreibung:
MCE Product type: Reference compound
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