FASN-IN-7 is a potent and orally active inhibitor of human Fatty Acid Synthase (FASN). FASN-IN-7 shows enzyme inhibition on full length FASN and the FASN KR domain with IC50 values of 28 and 54 nM. FASN-IN-7 effectively inhibits proliferation of multiple cancer cell types. FASN-IN-7 increases malonyl-CoA levels and decreases palmitate levels in tumor tissues[1].
Molekulargewicht:
493.60
CAS Nummer:
[1579514-16-1]
Formel:
C30H31N5O2
Target-Kategorie:
Fatty Acid Synthase (FASN)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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