CBPD-268 is a potent and orally active CBP/p300 PROTAC degrader with an DC50 value of 0.03 nM. CBPD-268 induces CBP/p300 degradation and inhibits cell growth. CBPD-268 shows antitumor activity. CBPD-268 has the potential for the research of AR-positive prostate cancer (Structure Note: Red, Androgen receptor degrader (HY-W248665A), Blue, CBP/p300 ligand (HY-161483), Black, Linker)[1].
Molekulargewicht:
819.90
Reinheit:
99.23
CAS Nummer:
[2832961-58-5]
Formel:
C44H47F2N9O5
Target-Kategorie:
Histone Acetyltransferase,PROTACs
Anwendungsbeschreibung:
Reference compound
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