AZ7976 (Compound 42) is a highly selective agonist for the Relaxin Family Peptide Receptor 1 (RXFP1) (pEC50 > 10.5). AZ7976 enhances RXFP1s cAMP signaling through an allosteric mechanism, thereby physiologically increasing heart rate. AZ7976 can be used in the field of cardiovascular disease research[1].
Molekulargewicht:
682.65
CAS Nummer:
[2813866-27-0]
Formel:
C30H33F7N2O6S
Target-Kategorie:
RXFP Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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