PPARdelta agonist 11, CAS [[2982696-04-6]] Preis auf Anfrage
Artikelnummer:
MCE-HY-162963
Hersteller Artikelnummer:
HY-162963
Alternativnummer:
MCE-HY-162963-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
PPARdelta agonist 11 (Compound 11) is a selective agonist for PPARdelta with an EC50 of 20 nM. PPARdelta agonist 11 reduces the levels of nitrite oxide (NO), proinflammatory cytokines TNFalpha and IL-6 in LPS (HY-D1056)-stimulated RAW264.7 cell, and exhibits anti-inflammatory efficacy via NF-kappaB pathway. PPARdelta agonist 11 exhibits good stability in human liver microsomes and plasma. PPARdelta agonist 11 ameliorates Carrageenan (HY-125474)-induced foot edema[1].
Molekulargewicht:
440.46
CAS Nummer:
[2982696-04-6]
Formel:
C19H15F3N2O3S2
Target-Kategorie:
PPAR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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