HTRA1-IN-1 (Compound 17) is a selective inhibitor for serine protease high temperature requirement A serine peptidase 1 (HTRA1), with IC50 of 13 nM. HTRA1-IN-1 is potential for ameliorating HTRA1-related diseases, such as age-related macular degeneration (AMD), osteoarthritis, and rheumatoid arthritis[1].
Molekulargewicht:
583.95
Reinheit:
96.96
CAS Nummer:
[3052552-04-9]
Formel:
C31H43BClN3O5
Target-Kategorie:
Ser/Thr Protease
Anwendungsbeschreibung:
Reference compound
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