CDK2 degrader 1, CAS [[3036604-59-5]]

Artikelnummer: MCE-HY-163814
Artikelname: CDK2 degrader 1, CAS [[3036604-59-5]]
Artikelnummer: MCE-HY-163814
Hersteller Artikelnummer: HY-163814
Alternativnummer: MCE-HY-163814-1MG,MCE-HY-163814-5MG,MCE-HY-163814-10MMX1ML,MCE-HY-163814-100MG,MCE-HY-163814-50MG,MCE-HY-163814-25MG,MCE-HY-163814-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
CDK2 degrader 1 (Compound 3) is a selective CDK2 molecular glue degrader with a Dmax (CDK2) of > 80% and a Ki (CRBN) > 1 µM. CDK2 degrader 1 binds to cereblon to induce ubiquitination and subsequent proteasomal degradation of the CDK2. CDK2 degrader 1 is used in the research of a wide range of cancers[1].
Molekulargewicht: 447.47
Reinheit: 99.74
CAS Nummer: [3036604-59-5]
Formel: C23H27F2N3O4
Target-Kategorie: CDK,Molecular Glues
Anwendungsbeschreibung: MCE Product type: Reference compound