SR-302, a chemical probe, is a potent and selectivity DDR/p38 inhibitor, with IC50 values of 0.125, 0.023 and 0.018 µM for p38alpha, DDR1 and DDR2, respectively. SR-302 can be used for the research of fibrotic disorders, such as renal and pulmonary fibrosis, atherosclerosis, and various forms of cancer[1].
Molekulargewicht:
622.78
Reinheit:
98.51
CAS Nummer:
[2771319-74-3]
Formel:
C32H42N6O5S
Target-Kategorie:
Discoidin Domain Receptor,p38 MAPK
Anwendungsbeschreibung:
MCE Product type: Reference compound
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