(R,R,S)-GAT107 is a fully agonistic positive modulator of alpha7 nicotinic receptors with significant biological activity. Its activity is entirely present in its (+)-isomer 1b, while (-)-isomer 1a does not affect its activity when used together. Studies have shown that (R,R,S)-GAT107 is the most potent ago-PAM for alpha7 nicotinic receptors currently known and has the potential for further in vivo evaluation[1].
Molekulargewicht:
405.31
CAS Nummer:
[1426240-47-2]
Formel:
C18H17BrN2O2S
Target-Kategorie:
Endogenous Metabolite
Anwendungsbeschreibung:
MCE Product type: Reference compound
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