5-HT6 inverse agonist 1, CAS [[2727088-38-0]] Preis auf Anfrage

Artikelnummer: MCE-HY-168333
Artikelname: 5-HT6 inverse agonist 1, CAS [[2727088-38-0]] Preis auf Anfrage
Artikelnummer: MCE-HY-168333
Hersteller Artikelnummer: HY-168333
Alternativnummer: MCE-HY-168333-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
5-HT6 inverse agonist 1 (Compound 33) is an antagonist for 5-HT6 receptor with a Ki of 23 nM and a Kb of 6.62 nM. 5-HT6 inverse agonist 1 inhibits the 5-HT6R mediated Cdk5 and mTOR signaling pathway. 5-HT6 inverse agonist 1 reduces tactile hypersensitivity in spinal nerve ligation (SNL)-induced rat model[1].
Molekulargewicht: 498.40
CAS Nummer: [2727088-38-0]
Formel: C22H22Cl2FN3O3S
Target-Kategorie: 5-HT Receptor,CDK,mTOR
Anwendungsbeschreibung: MCE Product type: Reference compound