sigma1 Receptor ligand 1 (compound 5I) is a sigma1 receptor ligand with a Ki of 3.9 nM. sigma1 Receptor ligand 1 has a high plasma protein binding (89%) and promising metabolic stability in the presence of mouse liver microsomes and NADPH. sigma1 Receptor ligand 1 can be utilized in neurological and cancer research[1].
Molekulargewicht:
352.47
Formel:
C22H28N2O2
Target-Kategorie:
Sigma Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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