MZ82, Ko 143 (HY-10010) derivative, is a ATP-binding cassette subfamily G member 2 (ABCG2/BCRP) inhibitor with the IC50 of ~23 nM. MZ82 not only shows greatly improved metabolic stability over Ko 143 (HY-10010) in liver microsomes but also in mice, and is able to penetrate into the brain[1].
Molekulargewicht:
431.53
CAS Nummer:
[2944457-11-6]
Formel:
C26H29N3O3
Target-Kategorie:
BCRP
Anwendungsbeschreibung:
MCE Product type: Reference compound
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