PROTAC HIF-1alpha degrader-1
Artikelnummer:
MCE-HY-168641
| Artikelname: |
PROTAC HIF-1alpha degrader-1 |
| Artikelnummer: |
MCE-HY-168641 |
| Hersteller Artikelnummer: |
HY-168641 |
| Alternativnummer: |
MCE-HY-168641-5MG,MCE-HY-168641-10MG,MCE-HY-168641-25MG,MCE-HY-168641-50MG |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| PROTAC HIF-1alpha degrader-1 (compound V2) is a potent hypoxia-inducible factor-1alpha (HIF-1alpha) PROTAC degrader with an IC50 value of 7.54 µM. PROTAC HIF-1alpha degrader-1 shows anti-proliferative activity. PROTAC HIF-1alpha degrader-1 decreases the HIF-1alpha protein expression. PROTAC HIF-1alpha degrader-1 induces apoptosis. (Pink: ligand for target protein (HY-111387), black: linker (HY-W013731), Blue: E3 ligase ligand (HY-112078))[1]. |
| Molekulargewicht: |
913.22 |
| Reinheit: |
98.02 |
| Formel: |
C51H72N6O7S |
| Target-Kategorie: |
Apoptosis,HIF/HIF Prolyl-Hydroxylase,PROTACs |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |