PROTAC HIF-1alpha degrader-1

Artikelnummer: MCE-HY-168641
Artikelname: PROTAC HIF-1alpha degrader-1
Artikelnummer: MCE-HY-168641
Hersteller Artikelnummer: HY-168641
Alternativnummer: MCE-HY-168641-5MG,MCE-HY-168641-10MG,MCE-HY-168641-25MG,MCE-HY-168641-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC HIF-1alpha degrader-1 (compound V2) is a potent hypoxia-inducible factor-1alpha (HIF-1alpha) PROTAC degrader with an IC50 value of 7.54 µM. PROTAC HIF-1alpha degrader-1 shows anti-proliferative activity. PROTAC HIF-1alpha degrader-1 decreases the HIF-1alpha protein expression. PROTAC HIF-1alpha degrader-1 induces apoptosis. (Pink: ligand for target protein (HY-111387), black: linker (HY-W013731), Blue: E3 ligase ligand (HY-112078))[1].
Molekulargewicht: 913.22
Reinheit: 98.02
Formel: C51H72N6O7S
Target-Kategorie: Apoptosis,HIF/HIF Prolyl-Hydroxylase,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound