PROTAC 20S proteasome subunit beta5 degrader 2 Preis auf Anfrage

Artikelnummer: MCE-HY-169135
Artikelname: PROTAC 20S proteasome subunit beta5 degrader 2 Preis auf Anfrage
Artikelnummer: MCE-HY-169135
Hersteller Artikelnummer: HY-169135
Alternativnummer: MCE-HY-169135-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC 20S proteasome subunit beta5 degrader 2 is a PROTAC degrader for 20S proteasome subunit beta5, with a DC50 of 0.16 µM. PROTAC 20S proteasome subunit beta5 degrader 2 inhibits the proliferation of cancer cell FaDu with IC50 of 0.23 µM. PROTAC 20S proteasome subunit beta5 degrader 2 exhibits antitumor efficacy in mice models[1]. (Pink: Ligand for target protein (HY-10227), Blue: Ligand for E3 ligase (HY-103596), Black: Linker (HY-Y1760))
Molekulargewicht: 845.74
Formel: C46H52BN5O10
Target-Kategorie: PROTACs,Proteasome
Anwendungsbeschreibung: MCE Product type: Reference compound