PROTAC 20S proteasome subunit beta5 degrader 2 Preis auf Anfrage
Artikelnummer:
MCE-HY-169135
Hersteller Artikelnummer:
HY-169135
Alternativnummer:
MCE-HY-169135-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
PROTAC 20S proteasome subunit beta5 degrader 2 is a PROTAC degrader for 20S proteasome subunit beta5, with a DC50 of 0.16 µM. PROTAC 20S proteasome subunit beta5 degrader 2 inhibits the proliferation of cancer cell FaDu with IC50 of 0.23 µM. PROTAC 20S proteasome subunit beta5 degrader 2 exhibits antitumor efficacy in mice models[1]. (Pink: Ligand for target protein (HY-10227), Blue: Ligand for E3 ligase (HY-103596), Black: Linker (HY-Y1760))
Molekulargewicht:
845.74
Formel:
C46H52BN5O10
Target-Kategorie:
PROTACs,Proteasome
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten