PKN3-IN-1 (compound 16) inhibits PKN3 (serine/threonine protein kinase 3) and GAK (cyclin G-associated kinase) with IC50 of 0.014 µM and Ki of 0.0044 µM respectively. PKN3-IN-1 is a potential tool compound to study the cell biology of PKN3 and its role in pancreatic and prostate cancer and T-cell acute lymphoblastic leukemia [1].
Molekulargewicht:
436.24
Reinheit:
98.97
CAS Nummer:
[2361545-75-5]
Formel:
C18H17IN2O3
Target-Kategorie:
PI3K
Anwendungsbeschreibung:
MCE Product type: Reference compound
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