alpha-Glucosidase-IN-79 (Compound 4d9) is a non-competitive alpha-Glucosidase inhibitor with an IC50 of 2.11 µM, which is more potent than existing alpha-Glucosidase inhibitors such as Acarbose (HY-B0089) (IC50 of 327.0 µM) and HXH8r (IC50 of 15.32 µM). alpha-Glucosidase-IN-79 is non-cytotoxic to human normal hepatocyte (LO2) cells and shows good metabolic stability in rat plasma. alpha-Glucosidase-IN-79 holds promise for research into type 2 diabetes[1].
Molekulargewicht:
414.47
Formel:
C21H22N2O5S
Target-Kategorie:
Glycosidase
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
