BU72 is a highly potent and long-acting agonist of µ and kappa opioid receptors, and also has a partial agonist effect on delta opioid receptors (EC50 values are 0.054, 0.033, and 0.58 nM, respectively). BU72 has a strong and long-lasting analgesic effect, which is mainly mediated by µ opioid receptors. BU72 has a long-lasting activity and can partially reverse the analgesic effect of morphine. BU72 can be used in the study of opioid dependence[1].
Molekulargewicht:
428.57
CAS Nummer:
[173265-76-4]
Formel:
C28H32N2O2
Target-Kategorie:
Opioid Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
