Enpp-1/3-IN-1 (Compound 5j) is an ENPP1/ENPP3 inhibitor, with IC50s of 0.59 µM (h-ENPP1) and 0.62 µM (h-ENPP3) respectively. Enpp-1/3-IN-1 also inhibits e5'NT (CD73) and TNAP with IC50s of 0.89 µM (h-e5'NT), 5.12 µM (r-e5'NT) and 1.68 µM (h-TNAP), respectively. Enpp-1/3-IN-1 can be used for cancer research[1].
Molekulargewicht:
398.36
Formel:
C17H13F3N2O4S
Target-Kategorie:
CD73,Phosphatase,Phosphodiesterase (PDE)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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