TRPV1 antagonist 10, CAS [[896584-55-7]] Preis auf Anfrage
Artikelnummer:
MCE-HY-172774
Hersteller Artikelnummer:
HY-172774
Alternativnummer:
MCE-HY-172774-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
TRPV1 antagonist 10 is an orally active and potent TRPV1 antagonist (IC50 = 33.06 nM), moderate to weak URAT1 (IC50 = 22.51 µM) and GLUT9 (60.25% at 50 µM) inhibitor. TRPV1 antagonist 10 has analgesic and urate-lowering effect. TRPV1 antagonist 10 can be studied for research in hyperuricemia and inflammatory pain[1].