PROTAC HDAC6 degrader 5 Preis auf Anfrage
Artikelnummer:
MCE-HY-174401
| Artikelname: |
PROTAC HDAC6 degrader 5 Preis auf Anfrage |
| Artikelnummer: |
MCE-HY-174401 |
| Hersteller Artikelnummer: |
HY-174401 |
| Alternativnummer: |
MCE-HY-174401-1UNIT |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| PROTAC HDAC6 degrader 5 (Compound 5a) is a highly selective PROTAC targeting HDAC6. PROTAC HDAC6 degrader 5 can effectively degrade HDAC6 in cells (IC50 = 43 nM). PROTAC HDAC6 degrader 5 reduces HDAC6 levels through proteasome- and CRBN-dependent mechanisms (Pink: Target protein ligand (HY-174408), Target protein ligand + linker (HY-174409), Blue: Pomalidomide (HY-10984), Pomalidomide 4-alkylC3-azide (HY-139341))[1]. |
| Molekulargewicht: |
898.96 |
| Formel: |
C47H50N10O9 |
| Target-Kategorie: |
HDAC,Ligands for E3 Ligase,PROTACs |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |