PROTAC FLT-3 degrader 5 Preis auf Anfrage

Artikelnummer: MCE-HY-175040
Artikelname: PROTAC FLT-3 degrader 5 Preis auf Anfrage
Artikelnummer: MCE-HY-175040
Hersteller Artikelnummer: HY-175040
Alternativnummer: MCE-HY-175040-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC FLT-3 degrader 5 is a FLT3 PROTAC degrader (DC50 = 1.2 nM). PROTAC FLT-3 degrader 5 functions as a molecular glue to degrade cereblon substrates GSPT1 and IKZF1/3. PROTAC FLT-3 degrader 5 exhibits antiproliferative activity against drug-resistant acute myeloid leukemia (AML) cells and is potentially useful in AML research. (Pink: FLT3/GSPT1/IKZF1/3 ligand: (HY-169374), Blue: Thalidomide: (HY-14658), Black: linker, Thalidomide + linker: (HY-W1123823))[1].
Molekulargewicht: 878.03
Formel: C46H59N11O7
Target-Kategorie: FLT3,IKZF Family,Molecular Glues,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound