MRT-7612 (Compound 4) is a cereblon-based tyrosine kinases molecular glue degrader. MRT-7612 significantly induces HCK and LYN degradation, with week efficacy on LCK. MRT-7612 can be used for cancers like chronic myeloid leukemia, autoimmune and chronic inflammatory diseases research[1].
Molekulargewicht:
444.48
Formel:
C25H24N4O4
Target-Kategorie:
Bcr-Abl,Molecular Glues,Src
Anwendungsbeschreibung:
MCE Product type: Reference compound
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