RJG-2051 is a selective covalent aldo-keto reductase family 1 member C3 (AKR1C3) inhibitor with an IC50 value of 13 nM. RJG-2051 interferes with the metabolic process of substrates such as androgens, estrogens, and prostaglandins by AKR1C3. RJG-2051 is promising for research of cancers[1].
Molekulargewicht:
509.62
CAS Nummer:
[2851993-77-4]
Formel:
C26H31N5O4S
Target-Kategorie:
Aldose Reductase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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