Nastorazepide (Standard), CAS [[209219-38-5]] Preis auf Anfrage
Artikelnummer:
MCE-HY-17617R
Hersteller Artikelnummer:
HY-17617R
Alternativnummer:
MCE-HY-17617R-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Nastorazepide (Standard) is the analytical standard of Nastorazepide. This product is intended for research and analytical applications. Nastorazepide (Z-360) is an orally active 1,5-benzodiazepine derivative and gastrin/CCK-2 receptor antagonist. Nastorazepide inhibits the specific binding of [3H]CCK-8 to the human CCK-2 receptor with a Ki value of 0.47 nM. Nastorazepide inhibits IL-1beta, ephrin B1, VEGF, and HIF-1alpha, reduces Akt and NR2B phosphorylation. Nastorazepide has antitumor activity against pancreatic cancer. Nastorazepide inhibits colorectal cancer liver metastasis and relieves pain[1][2][3][4][5][6][7].