Lumateperone-d4, CAS [[2102683-55-4]] Preis auf Anfrage
Artikelnummer:
MCE-HY-17637S2
Hersteller Artikelnummer:
HY-17637S2
Alternativnummer:
MCE-HY-17637S2-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Alternative Synonym:
ITI-007-d4
Lumateperone-d4 (ITI-007-d4) is deuterium labeled Lumateperone. Lumateperone (ITI-007) is an orally active 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone has anticancer activity and can also be used for the study of schizophrenia and bipolar depression[1][2][3].