PROTAC pan-KRAS degrader-1, CAS [[3043908-63-7]] Preis auf Anfrage
Artikelnummer:
MCE-HY-176489
Hersteller Artikelnummer:
HY-176489
Alternativnummer:
MCE-HY-176489-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
PROTAC pan-KRAS degrader-1 is a pan-KRAS PROTAC degrader for degrading different KRAS mutation types, such as G12D, G12C, G12V, and G13D. PROTAC pan-KRAS degrader-1 potently degrades KRAS mutation (G12D) in AGS cells, with a DC50 of 1.1 nM, Dmax of 95%. PROTAC pan-KRAS degrader-1 can be used to search diseases caused by KRAS mutation or amplification, especially cancers such as breast cancer, bladder cancer, gastric cancer, etc[1]. Pink: pan-KRAS ligand (HY-176490), Blue: VHL ligase ligand (HY-170353), Black: linker (HY-176491),
Molekulargewicht:
1192.38
CAS Nummer:
[3043908-63-7]
Formel:
C63H71F2N13O7S
Target-Kategorie:
PROTACs,Ras
Anwendungsbeschreibung:
MCE Product type: Reference compound
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