TG-2-IN-5 (Compound CP4d) is a reversible TG2 inhibitor with a Ki of 1.0 µM for human TG2. TG-2-IN-5 can be used to study diseases associated with upregulation of TG2-mediated acyl transfer, such as fibrosis and cancer[1].
Molekulargewicht:
379.33
CAS Nummer:
[1082605-61-5]
Formel:
C18H13N5O5
Target-Kategorie:
Glutaminase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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