Ciprokiren (Ro 44-9375) is a Renin inhibitor with IC50s of 0.07 and 0.65 nM for hRenin in buffer and plasma, respectively. Ciprokiren be applied transdermally with similar hemodynamic effects without decrease of plasma renin activity or plasma immunoreactive angiotensin II. Ciprokiren has antihypertensive efficacy and can be used for hypertension research[1].
Molekulargewicht:
729.93
CAS Nummer:
[143631-62-3]
Formel:
C37H55N5O8S
Target-Kategorie:
Renin
Anwendungsbeschreibung:
MCE Product type: Reference compound
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