SSTR3 agonist-1 TFA is a potent, orally active, and selective SSTR3 agnoist (EC50 =0.14 nM). SSTR3 agonist-1 TFA binds to SSTR3 receptor to inhibit cAMP activity. SSTR3 agonist-1 TFA decreases kidney weight and kidney cystic index (KCI) in a mouse model of autosomal dominant polycystic kidney disease (ADPKD). SSTR3 agonist-1 TFA can be used for ADPKD research[1].
Molekulargewicht:
733.67
Reinheit:
98.86
Formel:
C33H38F7N5O6
Target-Kategorie:
Somatostatin Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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