PROTAC CDK4/6/9 degrader 1, CAS [[3064994-97-1]] Preis auf Anfrage

Artikelnummer: MCE-HY-178452
Artikelname: PROTAC CDK4/6/9 degrader 1, CAS [[3064994-97-1]] Preis auf Anfrage
Artikelnummer: MCE-HY-178452
Hersteller Artikelnummer: HY-178452
Alternativnummer: MCE-HY-178452-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC CDK4/6/9 degrader 1 is a CDK4/6/9 PROTAC degrader. PROTAC CDK4/6/9 degrader 1 degrades CDK4, CDK6, and CDK9 in TNBC cells and inhibits TNBC cell proliferation. PROTAC CDK4/6/9 degrader 1 induces G1 phase arrest, promotes apoptosis, and suppresses cell migration and invasion in TNBC cells. PROTAC CDK4/6/9 degrader 1 can be used for the study of triple-negative breast cancer (TNBC). (Pink: CDK4/6/9 ligand (HY-168440), Blue: CRBN Ligand (HY-14658), Black: Linker (HY-178512), E3 ligase ligand-linker conjugate (HY-178515))[1].
Molekulargewicht: 955.11
CAS Nummer: [3064994-97-1]
Formel: C51H62N12O7
Target-Kategorie: Apoptosis,CDK,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound