CDD-1274 is an ERalpha (Estrogen receptor alpha) variant inhibitor. CDD-1274 induces proteasomal degradation of ERalpha variants in breast cancer cell lines and causes Y537S ERalpha degradation. CDD-1274 potently blocks ligand-dependent and ligand-independent ER signaling in endocrine-resistant breast cancer cells. CDD-1274 can be used for the study of breast cancer[1].
Molekulargewicht:
567.57
Formel:
C28H33F4N3O5
Target-Kategorie:
Estrogen Receptor/ERR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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