Dyrk1A-IN-15, CAS [[1448757-02-5]] Preis auf Anfrage

Artikelnummer: MCE-HY-179599
Artikelname: Dyrk1A-IN-15, CAS [[1448757-02-5]] Preis auf Anfrage
Artikelnummer: MCE-HY-179599
Hersteller Artikelnummer: HY-179599
Alternativnummer: MCE-HY-179599-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Dyrk1A-IN-15 is a selective, brain-penetrant and ATP-competitive Dyrk1A inhibitor with a IC50 of 19 nM. Dyrk1A-IN-15 displays high selectivity across a broad kinase panel (specific for DYRK kinases) with nanomolar potency. Dyrk1A-IN-15 impairs neurosphere self-renewal, cell invasion, and EGFR stability in vitro. Dyrk1A-IN-15 inhibits tumor growth and prolongs survival in vivo. Dyrk1A-IN-15 has potential for glioblastoma (GBM) research[1].
Molekulargewicht: 287.29
CAS Nummer: [1448757-02-5]
Formel: C14H9NO4S
Target-Kategorie: DYRK,EGFR
Anwendungsbeschreibung: MCE Product type: Reference compound