A2A/A3 agonist-1 is a dual A2A/A3 adenosine receptor agonist. A2A/A3 agonist-1 has a Ki value of 2.9 nM and an EC50 of 0.51 nM for hA2AAR. A2A/A3 agonist-1 has a Ki of 0.8 nM and an EC50 hA3AR. A2A/A3 agonist-1 possesses anti-inflammatory activity and can be used for the research of inflammatory diseases[1].
Molekulargewicht:
404.49
Formel:
C18H24N6O3S
Target-Kategorie:
Adenosine Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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