Cbz-QFR-kbt, CAS [[3086979-57-6]] Preis auf Anfrage
Artikelnummer:
MCE-HY-179708
Hersteller Artikelnummer:
HY-179708
Alternativnummer:
MCE-HY-179708-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Cbz-QFR-kbt is a ketone-based benzothiazole ketone inhibitor of TMPRSS2, with an IC50 value of 0.42 nM. Cbz-QFR-kbt also has inhibitory activity against Matriptase, Hepsin, HGFA, and Factor Xa, with IC50 values of 1, 1.3, 85, and 85 nM respectively. Cbz-QFR-kbt shows significant inhibitory effects against SARS-CoV-2 and H1N1 (IC50 = 60 nM). Cbz-QFR-kbt can be used in antiviral research[1].